Drug Design

Drug design, also known as rational drug design, is the process of creating new drugs based on the knowledge of the target and the interactions between the drug and the target. Drug design is a complex and extensive process that involves several steps such as target identification, lead discovery, lead optimization, and preclinical development. The first step in drug design is the identification of a specific target that is responsible for a particular disease. This target can be a protein or an enzyme that is involved in the disease process. Once the target is identified, the next step is to find a suitable lead compound that can interact with the target and modulate its activity. Lead discovery involves screening large libraries of compounds to find potential leads that can bind to the target. The lead compounds are then optimized to improve their potency, selectivity, and pharmacokinetic properties. Various computational and experimental techniques are used to optimize the lead compounds. Once the lead compounds have been optimized, they undergo preclinical development, which involves studies to determine their safety, efficacy, and pharmacokinetic properties. This includes animal studies, toxicology, and formulation development. Drug design is a critical process in the pharmaceutical industry as it is essential in discovering new drugs to treat a wide range of diseases. By using advanced pharmaceutical science and technology, drug design has become more efficient and effective in recent years, leading to the discovery of new drugs that have significantly improved patient outcomes.

← Journal of Advanced Pharmaceutical Science And Technology

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36 article(s) found

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Pattern of Use of Highly Active Antiretroviral Therapy Regimens and Pattern of Occurrence of Adverse Drug Reactions in an Indian Human Immunodeficiency Virus Positive Patients

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Evaluation of SterculiaUrens Gum as Novel Carrier for Oral Colon Targeted Drug Delivery System

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Current Status of Nonsteroidal Anti-Inflammatory Drugs in Colorectal Cancer Prevention

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Management of Absent Capsular Support with a new Intraocular Lens Design

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Synthesis and Assessment of a New Tetrahydrogeraniol Derivative as Penetration Enhancer for Transdermal Drug Delivery

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A Successful Vancomycin Treatment of Multidrug-Resistant MRSA-Associated Canine Pyoderma

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Trends and inducing factors for illicit drug use in Grenada: Epoch 2001 – 2009.

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Novel N-Pyrrolylcarboxylic Acid Derivative as a Potential New Analgesic and Anti-Inflammatory Drug

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Regulation of Expression of Reactive Oxygen Intermediates During Plasmodium Infection to Reduce Immunopathology Provides a Possible Antioxidant Adjuvant to Enhance Anti-Malarial Drug Therapy

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Storing Lesion-free Tooth Morphology for Biomorphic Dental Restoration Design

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Profile of Similarity of Electron Withdrawing Structure Towards Analgesic-Anti-Inflammatory Activity of The Novel Isatin Analogue: Design and Implementation of Phase I Drug Discovery

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Evaluation of Bacterial Population in the Saliva of Drug Addicts

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Drug Design Progress of In silico, In vitro and In vivo Researches

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5S Dashboard Design Principles for Self-Service Business Intelligence Tool Users

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Drug Abuse among Street Children

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The Pineal Hypothesis for Drug Dependence

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Why New Drugs, Treatments, and Medical Devices Still Needs to be Tested Clinically Before Making it Available in the Market?

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Design Support to steer Creative Wicked Problem Solving Processes with Knowledge Management and Artificial Intelligence

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Successful Cascade of Care and Cure HCV in 5382 Drugs Users: How Increase HCV Treatment by Outreach Care, Since Screening to Treatment

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Characterization of rpoB Gene Mutations Associated with Rifampicin Resistance in Multidrug Resistant Tuberculosis Patients Co-infected with HIV from Southern India.

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Lipid Assemblies as Tools for Drug Delivery

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Assessment of Self Medication Practice and Drugs Storage Among South Sudanese Community in Addis Ababa, Ethiopia

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Treatment of Dairy Industry Wastewater - Special Reference to Design of Aerated Lagoon

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By Design: Aligning Structure with Values to Impact Outcomes in a Public Utility Model

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Design of Stopwatch based on STC89C52 Single Chip Microcomputer

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A Review on Drug Design by the Application of Computer

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Risk Management: Emerging critical issues during the hospital administration of drug therapy

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The Design and Demonstrative Analysis of the Gas Turbine Operation’s Simulator

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A case of delayed allergy after cyanoacrylate closure of varicose veins, diagnosed by drug-induced lymphocyte stimulation test

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Human Immunodeficiency Virus Drug Resistance (HIVDR) and Baseline Characteristics among Antiretroviral Therapy (ART) experienced Children and Adolescents under the care of Chidamoyo Christian Hospital in Hurungwe, Zimbabwe

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Spirometric profile of people living with HIV on antiretroviral drugs in Abidjan

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Measuring Quality Change in the Market for Anti-Ulcer Drugs

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Call to Action: The Need for Adverse Drug Event (ADE) Standardization and Codification Through Improved ADE Definitions, Documentation and Mapping, as well as More Refined Medication Definitions

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Toxicology and Drug Safety Issues: A Review Article

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Characterization of People Receiving 2-Drug Regimens (2DR) for HIV Management in Italy

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